C. Robin Ganellin: search on Z-Library

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1

Modulation of GABAA receptors and inhibitory synaptic currents by the endogenous CNS sleep regulator cis-9,10-octadecenoamide (cOA)

George Lees, Michelle D. Edwards, Abdul A. Hassoni, C Robin Ganellin, Dimitrious Galanakis

Journal:

British Journal of Pharmacology

Year:

1998

Language:

english

File:

PDF, 460 KB

english, 1998

2

Inhibitors of Tripeptidyl Peptidase II. 3. Derivation of Butabindide by Successive Structure Optimizations Leading to a Potential General Approach to Designing Exopeptidase Inhibitors

Ganellin, C. Robin, Bishop, Paul B., Bambal, Ramesh B., Chan, Suzanne M. T., Leblond, Bertrand, Moore, Andrew N. J., Zhao, Lihua, Bourgeat, Pierre, Rose, Christiane, Vargas, Froylan, Schwartz, Jean-Ch

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 167 KB

english, 2005

3

Glossary of terms used in medicinal chemistry. Part II (IUPAC Recommendations 2013)

Buckle, Derek R., Erhardt, Paul W., Ganellin, C. Robin, Kobayashi, Toshi, Perun, Thomas J., Proudfoot, John, Senn-Bilfinger, Joerg

Journal:

Pure & Applied Chemistry

Year:

2013

Language:

english

File:

PDF, 193 KB

english, 2013

4

A Novel Series of (Phenoxyalkyl)imidazoles as Potent H 3 -Receptor Histamine Antagonists †

Ganellin, C. Robin, Fkyerat, Abdellatif, Bang-Andersen, Benny, Athmani, Salah, Tertiuk, Wasyl, Garbarg, Monique, Ligneau, Xavier, Schwartz, Jean-Charles

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 333 KB

english, 1996

5

Histamine and its receptors

Mike E Parsons, C Robin Ganellin

Journal:

British Journal of Pharmacology

Year:

2006

Language:

english

File:

PDF, 192 KB

english, 2006

6

Isocytosine H2-receptor histamine antagonists II. Synthesis and evaluation of biological activity at histamine H1- and H2-receptors of 5-(heterocyclyl)methylisocytosines

Thomas H Brown, Robert C Blakemore, Peter Blurton, Graham J Durant, C.Robin Ganellin, Michael E Parsons, Anthony C Rasmussen, D.Anthony Rawlings, Terence F Walker

Journal:

European Journal of Medicinal Chemistry

Year:

1989

Language:

english

File:

PDF, 771 KB

english, 1989

7

Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR)

Bhaskar C. Das, Ankanahlli V. Madhukumar, Jaime Anguiano, Sean Kim, Michael Sinz, Tatyana A. Zvyaga, Eoin C. Power, C. Robin Ganellin, Sridhar Mani

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 185 KB

english, 2008

8

On the Concept of a Bivalent Pharmacophore for SKCa Channel Blockers: Synthesis, Pharmacological Testing, and Radioligand Binding Studies on Mono-, Bis-, and Tris-quinolinium Compounds

Dimitrios Galanakis, C. Robin Ganellin, Philip M. Dunn, Donald H. Jenkinson

Journal:

Archiv der Pharmazie

Year:

1996

Language:

english

File:

PDF, 490 KB

english, 1996

9

ChemInform Abstract: Benzophenone Derivatives and Related Compounds as Potent Histamine H3-Receptor Antagonists and Potential PET/SPECT Ligands.

Astrid Sasse, Xavier Ligneau, Bassem Sadek, Sigurd Elz, Heinz H. Pertz, C. Robin Ganellin, Jean-Michel Arrang, Jean-Charles Schwartz, Walter Schunack, Holger Stark

Journal:

Year:

2001

File:

PDF, 34 KB

2001

10

Robin Ganellin gives his views on medicinal chemistry and drug discovery

C.Robin Ganellin

Journal:

Drug Discovery Today

Year:

2004

Language:

english

File:

PDF, 38 KB

english, 2004

11

Selective impairment of atrioventricular conduction by 2-(2-pyridyl)-ethylamine and 2-(2-thiazolyl)-ethylamine, two histamine H1-receptor agonists

Roberto Levi, C.Robin Ganellin, Geoffrey Allan, Howard J. Willens

Journal:

European Journal of Pharmacology

Year:

1975

Language:

english

File:

PDF, 307 KB

english, 1975

12

New Histamine H 3 -Receptor Ligands of the Proxifan Series: Imoproxifan and Other Selective Antagonists with High Oral in Vivo Potency †

Sasse, Astrid, Sadek, Bassem, Ligneau, Xavier, Elz, Sigurd, Pertz, Heinz H., Luger, Peter, Ganellin, C. Robin, Arrang, Jean-Michel, Schwartz, Jean-Charles, Schunack, Walter, Stark, Holger

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 156 KB

english, 2000

13

Introduction to Biological and Small Molecule Drug Research and Development || Preface

Robin Ganellin, C.

Year:

2013

Language:

english

File:

PDF, 27 KB

english, 2013

14

Analogue-based Drug Discovery (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || The History of Drospirenone

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 75 KB

english, 2006

15

Analogue-based Drug Discovery (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || Optimizing Antihypertensive Therapy by Angiotensin Receptor Blockers

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 105 KB

english, 2006

16

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || β-Adrenoceptor Agonists and Asthma

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 160 KB

english, 2010

17

The Synthesis and Some Pharmacological Actions of the Enantiomers of the K+-Channel Blocker Cetiedil

Craig J. Roxburgh, C. Robin Ganellin, Mark A. R. Shiner, David C. H. Benton, Philip M. Dunn, Yeshi Ayalew, Donald H. Jenkinson

Journal:

Journal of Pharmacy and Pharmacology

Year:

1996

Language:

english

File:

PDF, 758 KB

english, 1996

18

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Dipeptidyl Peptidase IV Inhibitors for the Treatment of Type 2 Diabetes

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 257 KB

english, 2010

19

Novel Partial Agonists for the Histamine H 3 Receptor with High in Vitro and in Vivo Activity †

Sasse, Astrid, Stark, Holger, Reidemeister, Sibylle, Hüls, Annette, Elz, Sigurd, Ligneau, Xavier, Ganellin, C. Robin, Schwartz, Jean-Charles, Schunack, Walter

Journal:

Journal of Medicinal Chemistry

Year:

1999

Language:

english

File:

PDF, 86 KB

english, 1999

20

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Paclitaxel and Epothilone Analogues, Anticancer Drugs

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 336 KB

english, 2010

21

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Clevudine, to Treat Hepatitis B Viral Infection

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 591 KB

english, 2010

22

The dipole moments of 1,3-dimethylthiourea, 1,3-dimethyl-2-cyanoguanidine and 1,1-bis-methylamino-2-nitroethene in a aqueous solution

Rodney C. Young, C. Robin Ganellin, Michael J. Graham, Edward H. Grant

Journal:

Year:

1982

Language:

english

File:

PDF, 402 KB

english, 1982

23

Isocytosine H2-receptor histamine antagonists I. Oxmetidine and related compounds

Thomas H Brown, Robert C Blakemore, Graham J Durant, John C Emmett, C.Robin Ganellin, Michael E Parsons, D.Anthony Rawlings, Terence F Walker

Journal:

European Journal of Medicinal Chemistry

Year:

1988

Language:

english

File:

PDF, 966 KB

english, 1988

24

Structural variations of 1-(4-(phenoxymethyl)benzyl)piperidines as nonimidazole histamine H3 receptor antagonists

Tibor Mikó, Xavier Ligneau, Heinz H Pertz, Jean-Michel Arrang, C Robin Ganellin, Jean-Charles Schwartz, Walter Schunack, Holger Stark

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 351 KB

english, 2004

25

Analogue-based Drug Discovery Volume c (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || Histamine H1 Blockers: From Relative Failures to Blockbusters within Series of Analogues

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 156 KB

english, 2006

26

Crystal and molecular structure of the histamine H2-receptor antagonists, N-methyl-N?-{2-[(5-methylimidazol-4-yl)methylthio]ethyl}thiourea (metiamide) and N-{2-[(imidazol-4-yl)methylthio]ethyl}-N?-methylthiourea (thiaburimamide)

Prout, Keith, Critchley, Stephen R., Ganellin, C. Robin, Mitchell, Robert C.

Journal:

Journal of the Chemical Society Perkin Transactions 2

Year:

1977

Language:

english

File:

PDF, 989 KB

english, 1977

27

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Tipranavir, a Non-Peptidic Protease Inhibitor for Multi-Drug Resistant HIV

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 354 KB

english, 2010

28

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Front Matter

Fischer, János, Ganellin, C. Robin

Year:

2010

File:

PDF, 118 KB

2010

29

Education of medicinal chemists in departments of medicinal chemistry (U.S.A.)

C. Robin Ganellin, Lester A. Mitscher, John G. Topliss

Journal:

Medicinal Research Reviews

Year:

1998

Language:

english

File:

PDF, 84 KB

english, 1998

30

Different antagonist binding properties of human and rat histamine H3 receptors

Holger Stark, Wolfgang Sippl, Xavier Ligneau, Jean-Michel Arrang, C.Robin Ganellin, Jean-Charles Schwartz, Walter Schunack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 720 KB

english, 2001

31

Analogue-based Drug Discovery Volume c (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || Corticosteroids: From Natural Products to Useful Analogues

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 161 KB

english, 2006

32

Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists

Young, Rodney C., Mitchell, Robert C., Brown, Thomas H., Ganellin, C. Robin, Griffiths, Robin, Jones, Martin, Rana, Kishore K., Saunders, David, Smith, Ian R.

Journal:

Journal of Medicinal Chemistry

Year:

1988

Language:

english

File:

PDF, 1.75 MB

english, 1988

33

[125I]iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain

Marie Korner, Marie-Louise Bouthenet, C Robin Ganellin, Monique Garbarg, Claude Gros, Robert J Ife, Nicole Sales, Jean-Charles Schwartz

Journal:

European Journal of Pharmacology

Year:

1986

Language:

english

File:

PDF, 741 KB

english, 1986

34

Synthesis and Structure−Activity Relationships of Cetiedil Analogues as Blockers of the Ca 2+ -Activated K + Permeability of Erythrocytes †

Roxburgh, Craig J., Ganellin, C. Robin, Athmani, Salah, Bisi, Alessandra, Quaglia, Wilma, Benton, David C. H., Shiner, Mark A. R., Malik-Hall, Misbah, Haylett, Dennis G., Jenkinson, Donald H.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 117 KB

english, 2001

35

Analogue-based Drug Discovery (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || Index

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 121 KB

english, 2006

36

Synthesis of pyridyl isosteres of thioperamide as H3-receptor histamine antagonists

Ganellin, C. Robin, Jayes, Dalia, Khalaf, Yasmin S., Tertiuk, Wasyl, Arrang, Jean-Michel, Defontaine, Nadia, Schwartz, Jean-Charles

Journal:

Collection of Czechoslovak Chemical Communications

Year:

1991

Language:

english

File:

PDF, 227 KB

english, 1991

37

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Application of Molecular Modeling in Analogue-Based Drug Discovery

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 222 KB

english, 2010

38

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Index

Fischer, János, Ganellin, C. Robin

Year:

2010

File:

PDF, 87 KB

2010

39

Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H3-receptor antagonists

Sven Graßmann, Bassem Sadek, Xavier Ligneau, Sigurd Elz, C.Robin Ganellin, Jean-Michel Arrang, Jean-Charles Schwartz, Holger Stark, Walter Schunack

Journal:

European Journal of Pharmaceutical Sciences

Year:

2002

Language:

english

File:

PDF, 223 KB

english, 2002

40

Analogue-Based Drug Discovery III (FISCHER:DRUG ANALOGS III O-BK) || Index

Fischer, János, Ganellin, C. Robin, Rotella, David P.

Year:

2012

Language:

english

File:

PDF, 67 KB

english, 2012

41

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Muscarinic Receptor Antagonists in the Treatment of COPD

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 248 KB

english, 2010

42

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) ||

Fischer, János, Ganellin, C. Robin

Year:

2010

File:

PDF, 5.30 MB

2010

43

Synthesis of Potent Non-imidazole Histamine H3-Receptor Antagonists

C. Robin Ganellin, Fabien Leurquin, Antonia Piripitsi, Jean-Michel Arrang, Monique Garbarg, Xavier Ligneau, Walter Schunack, Jean-Charles Schwartz

Journal:

Archiv der Pharmazie

Year:

1998

Language:

english

File:

PDF, 293 KB

english, 1998

44

10.1038/35048583

Arrang, Jean-Michel, Morisset, Séverine, Rouleau, Agnès, Ligneau, Xavier, Gbahou, Florence, Tardivel-Lacombe, Joël, Stark, Holger, Schunack, Walter, Ganellin, C. Robin

Journal:

Year:

2000

Language:

english

File:

PDF, 438 KB

english, 2000

45

Synthesis and Quantitative Structure−Activity Relationship of a Novel Series of Small Conductance Ca 2+ -Activated K + Channel Blockers Related to Dequalinium

Galanakis, Dimitrios, Davis, Carole A., Ganellin, C. Robin, Dunn, Philip M.

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 478 KB

english, 1996

46

Analogue-based Drug Discovery (FISCHER: ANALOGUE-BASED DRUG DISCOVERY O-BK) || Development of Opioid Receptor Ligands

Fischer, János, Ganellin, C. Robin

Year:

2006

Language:

english

File:

PDF, 153 KB

english, 2006

47

Analogue-Based Drug Discovery II (FISCHER:DRUG ANALOGS II O-BK) || Eplerenone: Selective Aldosterone Antagonist

Fischer, János, Ganellin, C. Robin

Year:

2010

Language:

english

File:

PDF, 507 KB

english, 2010

48

Search for Histamine H3 Receptor Ligands with Combined Inhibitory Potency at Histamine N-Methyltransferase: ω-Piperidinoalkanamine Derivatives.

Sven Grassmann, Joachim Apelt, Xavier Ligneau, Heinz H. Pertz, Jean-Michel Arrang, C. Robin Ganellin, Jean-Charles Schwartz, Walter Schunack, Holger Stark

Journal:

Year:

2005

File:

PDF, 15 KB

2005

49

Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BKCa)

Eoin C. Power, C. Robin Ganellin, David C.H. Benton

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 118 KB

english, 2006

50

Analogues and derivatives of ciproxifan, a novel prototype for generating potent histamine H3-receptor antagonists

Holger Stark, Xavier Ligneau, Bassem Sadek, C.Robin Ganellin, Jean-Michel Arrang, Jean-Charles Schwartz, Walter Schunack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 153 KB

english, 2000

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